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| 别名: | |||
|---|---|---|---|
| Cas号: | 1049741-81-2 | 物化性质: | |
| 分子式: | C16H18N2O2 · HCl | 熔点: | |
| 分子量: | 306.79 | 沸点: | |
| EINECS编号: | 密度: | ||
| MDL号: | MFCD08705321 | 储存条件: | 2-8°C |
| 技术规格说明书 | |||
| 货号 | 规格 | 可用库存 | 销售价(RMB) | 您的折扣价(RMB) | 数量 | 加入购物车 |
|---|---|---|---|---|---|---|
| C920930-5mg | ≥98% (HPLC), solid | 预计交期：8~10个工作日 | 1,707.00 | 加入购物车 |
| 用途: | Ciproxifan belongs to a novel chemical series of histamine H3-receptor antagonists. In vitro, it behaved as a competitive antagonist at the H3 autoreceptor controlling 3H histamine release from synaptosomes and displayed similar Ki values (0.5-1.9 nM) at the H3 receptor controlling the electrically-induced contraction of guinea pig ileum or at the brain H3 receptor labeled with 125I-iodoproxyfan. Ciproxifan appears to be an orally bioavailable, extremely potent and selective H3-receptor antagonist whose vigilance- and attention-promoting effects are promising for therapeutic applications in aging disorders. |
|---|---|
| 储存条件: | 2-8°C |
| 颜色: | 固体 |
